药理:Protein kinase C (PKC) inhibitor. Inhibits PKCΙ and PKCζ; (IC50 values are 132 and 639 nM, respectively). Restores polarized morphogenesis in oncogene expressing MDCK cells, decreases colony formation in HeLa cells and inhibits lethal giant larvae 2 (LLGL2) phosphorylation.
溶解度:water|48.85|100|DMSO|48.85|100|